Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_06385
Ion Channel
Sodium channel protein type 4 subunit alpha
Peptide Function
Antagonist
Gene Name
SCN4A
Activity Data (nM)
IC50
69 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
RDCCTXXKKCKDRQCKXQRCCA
Peptide UniProt Accession
Not available
UniParc
Not available
Peptide Synonyms/Alias
[Geographutoxin I; mu-conotoxin GIIIA; 129129-65-3; mu-Conotoxin G IIIA; 86394-16-3; CHEMBL4562161; Conotoxin G IIIA; .mu.-Conotoxin G IIIA; UNII-0C5T02KI0E; 0C5T02KI0E; mu-Conotoxin G IIIA (reduced); DTXSID101339126; BDBM50520482; L-Alaninamide; L-arginyl-L-alpha-aspartyl-L-cysteinyl-L-cysteinyl-L-threonyl-(4R)-4-hydroxy-L-prolyl-(4R)-4-hydroxy-L-prolyl-L-lysyl-L-lysyl-L-cysteinyl-L-lysyl-L-alpha-aspartyl-L-arginyl-L-glutaminyl-L-cysteinyl-L-lysyl-(4R)-4-hydroxy-L-prolyl-l]
Peptide Species
Not specified
Peptide Name
Not available
CAS Number
129129-65-3
Experimental Conditions
pH
pH 7.4
Holding Potential (mV)
−70 mV
Temperature
18 °C
Test Method
Patch-clamping
Test Species
Xenopus laevis oocyte
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
VGSCs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)
References & Disease Information
Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available